phaclofen [Ligand Id: 1091] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1255941 (Phaclofen)
  • GABAB receptor in Human [GtoPdb: 242]
  • GABAB receptor in Rat [GtoPdb: 242]
  • This target only has 1 pki data point
1 CHEMBL1255941_lig_chart_1 GABAB receptor HumanRat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GABAB receptor in Human [GtoPdb: 242]
GtoPdb - - 3.9 pKi - - - Br. J. Pharmacol. (2000) 131: 1050-4 [PMID:11082110]
GABAB receptor in Rat [GtoPdb: 242]
GtoPdb - - 4.1 pIC50 - - - Pharmacol. Rev. (2002) 54: 247-64 [PMID:12037141]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]