HTL22562 [Ligand Id: 11113] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • CGRP receptor in Human [GtoPdb: 48]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CGRP receptor in Human [GtoPdb: 48]
GtoPdb Human CGRP receptors (consisting of CLR and RAMP1) were expressed in insect Sf21 cells. Dissociation constant was determined in a radioligand binding assay using hCGRPR-containing membrane homegenates and 3H-telcagepant as tracer. - 10.5 pKi - - - J Med Chem (2020) 63: 7906-7920 [PMID:32558564]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.