compound 5 [Stecula et al., 2020] [Ligand Id: 11155] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2409288
  • N-acetyltransferase 8 like in Human [GtoPdb: 3144] [UniProtKB: Q8N9F0]
  • This target only has 1 pki data point
  • 6.4
1 CHEMBL2409288_lig_chart_1 N-acetyltransferase 8 like Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
N-acetyltransferase 8 like in Human [GtoPdb: 3144] [UniProtKB: Q8N9F0]
GtoPdb - - 6.4 pKi 400 nM Ki Journal of Medicinal Chemistry (2020) :

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]