BIIB091 [Ligand Id: 11203] activity data from GtoPdb

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  • Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
GtoPdb Measuring inhibition of substrate peptide phosphorylation in the presence of active BTK enzyme, ATP, and inhibitor. - 9 pIC50 <1 nM IC50 WO2018191577A1. Benzoazepine analogs as inhibiting agents for bruton's tyrosine kinase (2018)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.