LYS006 [Ligand Id: 11205] activity data from GtoPdb

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  • Leukotriene A4 hydrolase in Human [GtoPdb: 1395] [UniProtKB: P09960]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 Leukotriene A4 hydrolase Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Leukotriene A4 hydrolase in Human [GtoPdb: 1395] [UniProtKB: P09960]
GtoPdb Inhibition of enzyme activity determined in a fluorescence assay using a 7-amino-4-methylcoumarin (AMC) arginine derivative (Arg-AMC) as a surrogate substrate for LTA4H. - 8.7 pIC50 2 nM IC50 WO2015092740A1. Heteroaryl butanoic acid derivatives as lta4h inhibitors (2015)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.