C3a receptor agonist [Ligand Id: 11252] activity data from GtoPdb

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  • C3a receptor in Human [GtoPdb: 31] [UniProtKB: Q16581]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
C3a receptor in Human [GtoPdb: 31] [UniProtKB: Q16581]
GtoPdb IC50 determined in a radioligand displacement assay; displacing [125I]C3a from hC3a receptor expressed in HMC1 cells co-expressing aequorin. - 6.1 pIC50 794 nM IC50 Bioorg Med Chem Lett (2007) 17: 3262-5 [PMID:17459702]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.