compound 73 [WO2017106607A1] [Ligand Id: 11307] activity data from GtoPdb

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  • TLR7 in Human [GtoPdb: 1757] [UniProtKB: Q9NYK1]
  • This target only has 0 pki data point
1 _lig_chart_1 TLR7 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TLR7 in Human [GtoPdb: 1757] [UniProtKB: Q9NYK1]
GtoPdb Inhibition of activation of a TLR7/NFkB reporter in HEK293 cells (binned value). - 6 pIC50 <1000 nM IC50 WO2017106607A1. Polycyclic tlr7/8 antagonists and use thereof in the treatment of immune disorders (2017)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.