M4205 [Ligand Id: 11510] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| platelet derived growth factor receptor alpha in Human [GtoPdb: 1803] [UniProtKB: P16234] | ||||||||
| GtoPdb | Biochemical inhibitory potency | - | 7.3 | pIC50 | 50 | nM | IC50 | J Med Chem (2023) 66: 2386-2395 [PMID:36728508] |
| platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619] | ||||||||
| GtoPdb | Biochemical inhibitory potency | - | 8.59 | pIC50 | 2.6 | nM | IC50 | J Med Chem (2023) 66: 2386-2395 [PMID:36728508] |
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | - | - | 7.36 | pIC50 | 44 | nM | IC50 | J Med Chem (2023) 66: 2386-2395 [PMID:36728508] |
| colony stimulating factor 1 receptor in Human [GtoPdb: 1806] [UniProtKB: P07333] | ||||||||
| GtoPdb | Biochemical inhibitory potency | - | 8.26 | pIC50 | 5.5 | nM | IC50 | J Med Chem (2023) 66: 2386-2395 [PMID:36728508] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
