ASTX029 [Ligand Id: 11727] activity data from GtoPdb

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  • mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
GtoPdb - - 8.57 pIC50 2.7 nM IC50 J Med Chem (2021) 64: 12286-12303 [PMID:34387469]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.