ceperognastat [Ligand Id: 11953] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| O-GlcNAcase in Human [GtoPdb: 3101] [UniProtKB: O60502] | ||||||||
| GtoPdb | Inhibition of OGA enzyme activity in vitro | - | 8.63 | pIC50 | 2.36 | nM | IC50 | WO2018140299A1. N-[4-fluoro-5-[[(2s,4s)-2-methyl-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-1-piperidyl]methyl]thiazol-2-yl]acetamide as oga inhibitor (2018) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
