allosteric modulator 33 [PMID: 35878399] [Ligand Id: 12071] activity data from GtoPdb

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  • Protein kinase G (PKG) 1 in Human [GtoPdb: 1492] [UniProtKB: Q13976]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Protein kinase G (PKG) 1 in Human [GtoPdb: 1492] [UniProtKB: Q13976]
GtoPdb Kinase activity determined for partially activated recombinant hPKG1α (with cGMP at EC20 concentration) - 6.28 pEC50 520 nM EC50 J Med Chem (2022) 65: 10318-10340 [PMID:35878399]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.