BMS-986339 [Ligand Id: 12109] activity data from GtoPdb

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  • Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Farnesoid X receptor in Human [GtoPdb: 603] [UniProtKB: Q96RI1]
GtoPdb Dtermined by measuring the transcriptional activity of FXR using an FXR-LBD/Gal4 luciferase reporter system - 7.47 pEC50 34 nM EC50 J Med Chem (2022) 65: 8948-8960 [PMID:35704802]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.