LSZ102 [Ligand Id: 12145] activity data from GtoPdb

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  • Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
GtoPdb Measuring inhibition of ER-mediated gene transcription in a luciferase reporter assay - 9.52 pIC50 0.3 nM IC50 J Med Chem (2018) 61: 2837-2864 [PMID:29562737]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.