JNJ-64264681 [Ligand Id: 12239] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BLK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 1940] [UniProtKB: P51451] | ||||||||
| GtoPdb | - | - | 5.5 | pIC50 | 3130 | nM | IC50 | J Med Chem (2022) 65: 14326-14336 [PMID:36314537] |
| BMX non-receptor tyrosine kinase in Human [GtoPdb: 1942] [UniProtKB: P51813] | ||||||||
| GtoPdb | - | - | 6.76 | pIC50 | 172 | nM | IC50 | J Med Chem (2022) 65: 14326-14336 [PMID:36314537] |
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | - | - | 7.31 | pKi | 48.5 | nM | Ki | J Med Chem (2022) 65: 14326-14336 [PMID:36314537] |
| GtoPdb | - | - | 6.25 | pIC50 | 558 | nM | IC50 | J Med Chem (2022) 65: 14326-14336 [PMID:36314537] |
| tec protein tyrosine kinase in Human [GtoPdb: 2238] [UniProtKB: P42680] | ||||||||
| GtoPdb | - | - | 6.52 | pIC50 | 303 | nM | IC50 | J Med Chem (2022) 65: 14326-14336 [PMID:36314537] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
