VU0486846 [Ligand Id: 12305] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229] | ||||||||
| GtoPdb | Agonist potency | - | 5.4 | pEC50 | 4000 | nM | EC50 | ACS Chem Neurosci (2018) 9: 2274-2285 [PMID:29701957] |
| GtoPdb | PAM potency | - | 6.51 | pEC50 | 310 | nM | EC50 |
ACS Chem Neurosci (2018) 9: 2274-2285 [PMID:29701957]; Bioorg Med Chem Lett (2018) 28: 2175-2179 [PMID:29754948] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
