emzeltrectinib [Ligand Id: 12377] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| neurotrophic receptor tyrosine kinase 1 in Human [GtoPdb: 1817] [UniProtKB: P04629] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | <1 | nM | IC50 | WO2018077246A1. Amino pyrazolopyrimidine compound used as neurotrophic factor tyrosine kinase receptor inhibitor (2018) |
| neurotrophic receptor tyrosine kinase 2 in Human [GtoPdb: 1818] [UniProtKB: Q16620] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | <1 | nM | IC50 | WO2018077246A1. Amino pyrazolopyrimidine compound used as neurotrophic factor tyrosine kinase receptor inhibitor (2018) |
| neurotrophic receptor tyrosine kinase 3 in Human [GtoPdb: 1819] [UniProtKB: Q16288] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | <1 | nM | IC50 | WO2018077246A1. Amino pyrazolopyrimidine compound used as neurotrophic factor tyrosine kinase receptor inhibitor (2018) |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 7 | pIC50 | >100 | nM | IC50 | WO2018077246A1. Amino pyrazolopyrimidine compound used as neurotrophic factor tyrosine kinase receptor inhibitor (2018) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
