fulzerasib [Ligand Id: 12393] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| KRAS in Human [GtoPdb: 2824] [UniProtKB: P01116] | ||||||||
| GtoPdb | HTRF assay detecting repacement of GDP by GTP on the KRASG12C protein catalyzed by SOS1 | - | 7.6 | pIC50 | 25 | nM | IC50 | WO2021083167A1. Substituted heterocyclic fused cyclic compound, preparation method therefor and pharmaceutical use thereof (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
