ChEMBL ligand: CHEMBL4105357
TAS2R16/Taste receptor type 2 member 16 in Human [ChEMBL: CHEMBL3309106] [GtoPdb: 669] [UniProtKB: Q9NYV7] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
TAS2R16/Taste receptor type 2 member 16 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3309106] [GtoPdb: 669] [UniProtKB: Q9NYV7]
GtoPdb	-	-	2.96	pEC50	1100000	nM	EC50	Nat Genet (2002) 32: 397-401 [PMID:12379855]
ChEMBL	Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio in presence of (E)-4-(2,2,3-trimethylcyclopent-3-enyl)but-2-enoic acid by Fluo-4 dye based FLIPR assay	F	6.6	pEC50	250	nM	EC50	US-8187822-B2. Methods to identify modulators (null)
ChEMBL	Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio by Fluo-4 dye based FLIPR assay	F	6.68	pEC50	210	nM	EC50	US-8187822-B2. Methods to identify modulators (null)

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]