GLPG2534 [Ligand Id: 12510] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • interleukin 1 receptor associated kinase 4 in Human [GtoPdb: 2045] [UniProtKB: Q9NWZ3]
  • interleukin 1 receptor associated kinase 4 in Mouse [GtoPdb: 2045] [UniProtKB: Q8R4K2]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
interleukin 1 receptor associated kinase 4 in Human [GtoPdb: 2045] [UniProtKB: Q9NWZ3]
GtoPdb Enzyme inhibition determined in a biochemical assay - 8.19 pIC50 6.4 nM IC50 Sci Transl Med (2023) 15: eabj3289 [PMID:36791209]
interleukin 1 receptor associated kinase 4 in Mouse [GtoPdb: 2045] [UniProtKB: Q8R4K2]
GtoPdb Enzyme inhibition determined in a biochemical assay - 8.46 pIC50 3.5 nM IC50 Sci Transl Med (2023) 15: eabj3289 [PMID:36791209]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.