nerandomilast [Ligand Id: 12518] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphodiesterase 4A in Human [GtoPdb: 1300] [UniProtKB: P27815] | ||||||||
| GtoPdb | Inhibition of PDE4A in vitro. | - | 6.61 | pIC50 | 248 | nM | IC50 | Front Pharmacol (2022) 13: 838449 [PMID:35517783] |
| phosphodiesterase 4B in Human [GtoPdb: 1301] [UniProtKB: Q07343] | ||||||||
| GtoPdb | Inhibition of PDE4B2 in vitro. | - | 8 | pIC50 | 10 | nM | IC50 | Front Pharmacol (2022) 13: 838449 [PMID:35517783] |
| phosphodiesterase 4D in Human [GtoPdb: 1303] [UniProtKB: Q08499] | ||||||||
| GtoPdb | Inhibition of PDE4D2 in vitro. | - | 7.04 | pIC50 | 91 | nM | IC50 | Front Pharmacol (2022) 13: 838449 [PMID:35517783] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
