ChEMBL ligand: CHEMBL438 (Mesulfa, Methypyrimal, NSC-27259, Sulfamerazina, Sulfamerazine, Sulfamerazine component of lantrisul, Sulfamerazine component of neotrizine, Sulfamerazine component of sulfaloid, Sulfamerazine component of sulfonamides duplex, Sulfamerazine component of sulfose, Sulfamerazine component of terfonyl, Sulfamerazine component of triple sulfoid, Sulfamerazine (trisulfapyrimidines), Sulfamerazine (trisulfapyrimidines) component of neotrizine, Sulfamerazine (trisulfapyrimidines) component of terfonyl, Sulfamethyldiazine, Sulphamerazine, Sumedin, Trisulfapyrimidines (sulfamerazine))

Plasmodium falciparum [ChEMBL: CHEMBL364] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
Plasmodium falciparum (target type: ORGANISM) [ChEMBL: CHEMBL364]
ChEMBL	Antiplasmodial activity against Plasmodium falciparum 3D7 infected in RBCs by firefly luciferase reporter gene assay	F	8.22	pIC50	6	nM	IC50	Antimicrob Agents Chemother (2010) 54: 3597-3604 [PMID:20547797]

ChEMBL data shown on this page come from version 36:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]