MMP13 tracer [18F]5j [Ligand Id: 12669] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| MMP8 in Human [GtoPdb: 1632] [UniProtKB: P22894] | ||||||||
| GtoPdb | - | - | 5.92 | pIC50 | 1200 | nM | IC50 | J Med Chem (2023) 66: 6682-6696 [PMID:37158732] |
| MMP10 in Human [GtoPdb: 1634] [UniProtKB: P09238] | ||||||||
| GtoPdb | - | - | 5.51 | pIC50 | 3100 | nM | IC50 | J Med Chem (2023) 66: 6682-6696 [PMID:37158732] |
| MMP13 in Human [GtoPdb: 1637] [UniProtKB: P45452] | ||||||||
| GtoPdb | Inhibitor potency against human recombinant MMP13, determined using the fluorogenic substrate Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 | - | 7.8 | pIC50 | 16 | nM | IC50 | J Med Chem (2023) 66: 6682-6696 [PMID:37158732] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
