STX-478 [Ligand Id: 12903] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | Affinity for wild type PI3Kα | - | 7.15 | pKd | 70 | nM | Kd | Cancer Discov (2023) 13: 2432-2447 [PMID:37623743] |
| GtoPdb | Affinity for PI3Kα with the H1047R mutation | - | 8.33 | pKd | 4.7 | nM | Kd | Cancer Discov (2023) 13: 2432-2447 [PMID:37623743] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
