biKEAP1 [Ligand Id: 13066] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| kelch like ECH-associated protein 1 in Human [GtoPdb: 2757] [UniProtKB: Q14145] | ||||||||
| GtoPdb | Determined in a fluorescence polarization (FP) assay, measuring displacement of a NRF2 ETGE motif derived peptide from KEAP1 Kelch domain | - | 8.07 | pIC50 | 8.49 | nM | IC50 | Cell Chem Biol (2024) 31: 1188-1202.e10 [PMID:38157852] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
