C3TD879 [Ligand Id: 13171] activity data from GtoPdb

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  • citron rho-interacting serine/threonine kinase in Human [GtoPdb: 1509] [UniProtKB: O14578]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
citron rho-interacting serine/threonine kinase in Human [GtoPdb: 1509] [UniProtKB: O14578]
GtoPdb Binding affinity - 8 pKd <10 nM Kd J Med Chem (2024) 67: 2631-2666 [PMID:38330278]
GtoPdb Catalytic inhibition in a biochemical assay. - 7.92 pIC50 12 nM IC50 J Med Chem (2024) 67: 2631-2666 [PMID:38330278]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.