rentosertib [Ligand Id: 13279] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| TRAF2 and NCK interacting kinase in Human [GtoPdb: 2244] [UniProtKB: Q9UKE5] | ||||||||
| GtoPdb | Binding affinity determined by surface plasmon resonance assay. | - | 8.36 | pKd | 4.32 | nM | Kd | Nat Biotechnol (2025) 43: 63-75 [PMID:38459338] |
| GtoPdb | - | - | 7.51 | pIC50 | 31 | nM | IC50 | Nat Biotechnol (2025) 43: 63-75 [PMID:38459338] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
