Teleocidin B4 [Ligand Id: 13408] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL417692 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| protein kinase C delta/Protein kinase C delta in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2996] [GtoPdb: 1485] [UniProtKB: Q05655] | ||||||||
| ChEMBL | Displacement of [3H]PDBu from recombinant Protein kinase C delta | B | 9.49 | pKi | 0.32 | nM | Ki | J Med Chem (1998) 41: 1476-1496 [PMID:9554881] |
| protein kinase C eta/Protein kinase C eta in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4992] [GtoPdb: 1487] [UniProtKB: P23298] | ||||||||
| ChEMBL | Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C eta | B | 10 | pKi | 0.1 | nM | Ki | Bioorg Med Chem Lett (1996) 6: 353-356 |
| protein kinase C gamma/Protein kinase C gamma in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3604] [GtoPdb: 1484] [UniProtKB: P63319] | ||||||||
| ChEMBL | Inhibition of [3H]- PDBu binding to peptide C, rat brain PKC gamma | B | 8.7 | pKi | 2 | nM | Ki | Bioorg Med Chem Lett (1996) 6: 353-356 |
ChEMBL data shown on this page come from version 35:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
