DA-302168S [Ligand Id: 13870] activity data from GtoPdb

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  • GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220]
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  • Kv11.1 in Human [GtoPdb: 572] [UniProtKB: Q12809]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220]
GtoPdb Determined using a luciferase assay in HEK293 cells expressing hGLP-1R - 8.88 pEC50 1.32 nM EC50 J Med Chem (2025) : [PMID:40257122]
Kv11.1 in Human [GtoPdb: 572] [UniProtKB: Q12809]
GtoPdb - - 4.52 pIC50 >30000 nM IC50 J Med Chem (2025) : [PMID:40257122]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.