compound 1 [PMID: 40415551] [Ligand Id: 13928] activity data from GtoPdb

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  • cathepsin B in Human [GtoPdb: 2343] [UniProtKB: P07858]
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  • cathepsin L in Human [GtoPdb: 2351] [UniProtKB: P07711]
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  • CoV 3C-like (main) protease in SARS-CoV-2 [GtoPdb: 3111]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cathepsin B in Human [GtoPdb: 2343] [UniProtKB: P07858]
GtoPdb - - 6.36 pIC50 436 nM IC50 J Med Chem (2025) : [PMID:40415551]
cathepsin L in Human [GtoPdb: 2351] [UniProtKB: P07711]
GtoPdb - - 7.54 pIC50 28.8 nM IC50 J Med Chem (2025) : [PMID:40415551]
CoV 3C-like (main) protease in SARS-CoV-2 [GtoPdb: 3111]
GtoPdb - - 8.61 pIC50 2.45 nM IC50 J Med Chem (2025) : [PMID:40415551]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.