AZD0233 [Ligand Id: 14193] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CX3CR1 in Human [GtoPdb: 74] [UniProtKB: P49238] | ||||||||
| GtoPdb | Measuring displacement of [3H]ADZ8797 in a competition binding assay | - | 7.28 | pIC50 | 52 | nM | IC50 | WO2024083933A1. 2,4,6-trisubstituted 1,3,5-triazines as modulators of cx3cr1 (2024) |
| GtoPdb | Measuring antagonism of β-arrestin recruitment | - | 7 | pEC50 | 100 | nM | EC50 | WO2024083933A1. 2,4,6-trisubstituted 1,3,5-triazines as modulators of cx3cr1 (2024) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
