AJ-292 [Ligand Id: 14267] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ADGRL2 in Human [GtoPdb: 207] [UniProtKB: O95490] | ||||||||
| GtoPdb | Binding affinity determined in HEK293 cells transfected with ADGRL2-Nluc, competitively displacing FITC-conjugated Stachel sequence peptide | - | 7.68 | pKi | 21.1 | nM | Ki | Cell Reports (2025) 44: 116519 |
| GtoPdb | Measuring antagonism of force-induced ADGRL2 Gs activation (cAMP accumulation) in ADGRL2-overexpressing HEK293 cells | - | 7.68 | pIC50 | 20.8 | nM | IC50 | Cell Reports (2025) 44: 116519 |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
