relcobatinib [Ligand Id: 14371] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ABL proto-oncogene 1, non-receptor tyrosine kinase in Human [GtoPdb: 1923] [UniProtKB: P00519] | ||||||||
| GtoPdb | Inhibition of ABL1T3151 in a biochemical assay | - | 7.36 | pIC50 | 43.5 | nM | IC50 | WO2022076975A1. 5- and 6-azaindole compounds for inhibition of bcr-abl tyrosine kinases (2022) |
| GtoPdb | Inhibition of WT ABL1 in a biochemical assay | - | 7.9 | pIC50 | 12.7 | nM | IC50 | WO2022076975A1. 5- and 6-azaindole compounds for inhibition of bcr-abl tyrosine kinases (2022) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
