BHV-2100 [Ligand Id: 14467] activity data from GtoPdb

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  • TRPM3 in Mouse [GtoPdb: 495]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPM3 in Mouse [GtoPdb: 495]
GtoPdb Measuring antagonism of pregnenolone-mediated calcium influx via mTRPM3α2 in HEK293 cells, monitored with the calcium-responsive fluorescent dye Fluor-4 AM - 6 pIC50 <1000 nM IC50 US12209081B2. Heterocycle derivatives for treating TRPM3 mediated disorders (2025)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.