ChEMBL ligand: CHEMBL192359 (AC-7954)
UT receptor/Urotensin II receptor in Human [ChEMBL: CHEMBL3764] [GtoPdb: 365] [UniProtKB: Q9UKP6] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
UT receptor/Urotensin II receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3764] [GtoPdb: 365] [UniProtKB: Q9UKP6]
GtoPdb	-	-	6.6	pKi	-	-	-	J Med Chem (2002) 45: 4950-3 [PMID:12408704]; Bioorg Med Chem (2005) 13: 3057-68 [PMID:15781415]
ChEMBL	Activity against human urotensin-2 receptor expressed in NIH3T3 cells	B	5.95	pEC50	1122.02	nM	EC50	J. Med. Chem. (2006) 49: 2232-2240 [PMID:16570919]
ChEMBL	Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT assay	F	5.95	pEC50	>=1122.02	nM	EC50	Bioorg. Med. Chem. (2009) 17: 4657-4665 [PMID:19481466]
ChEMBL	Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT assay	F	5.95	pEC50	1122.02	nM	EC50	Bioorg. Med. Chem. (2010) 18: 4844-4854 [PMID:20570157]
ChEMBL	Agonist activity for human Urotensin 2 receptor	F	6.52	pEC50	300	nM	EC50	J. Med. Chem. (2005) 48: 2480-2492 [PMID:15801838]
ChEMBL	Agonist activity at human urotensin 2 expressed in CHO cells by FLIPR	F	6.6	pEC50	250	nM	EC50	J. Med. Chem. (2010) 53: 2695-2708 [PMID:20043680]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]