d(CH2)5[Tyr(Me)2,Thr4,Tyr-NH29]OVT [Ligand Id: 2221] activity data from GtoPdb

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  • V1A receptor in Human [GtoPdb: 366] [UniProtKB: P37288]
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  • V1B receptor in Human [GtoPdb: 367] [UniProtKB: P47901]
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  • V2 receptor in Human [GtoPdb: 368] [UniProtKB: P30518]
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  • OT receptor in Human [GtoPdb: 369] [UniProtKB: P30559]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
V1A receptor in Human [GtoPdb: 366] [UniProtKB: P37288]
GtoPdb - - 8.4 pKi - - - Endocrinology (1997) 138: 4109-22 [PMID:9322919];
J Pept Sci (2005) 11: 593-608 [PMID:15880385]
V1B receptor in Human [GtoPdb: 367] [UniProtKB: P47901]
GtoPdb - - 5 pKi - - - Endocrinology (1997) 138: 4109-22 [PMID:9322919]
V2 receptor in Human [GtoPdb: 368] [UniProtKB: P30518]
GtoPdb - - 6 pKi - - - Endocrinology (1997) 138: 4109-22 [PMID:9322919];
Kidney Int (2000) 58: 1613-22 [PMID:11012895]
OT receptor in Human [GtoPdb: 369] [UniProtKB: P30559]
GtoPdb - - 10 pKi - - - J Pept Sci (2005) 11: 593-608 [PMID:15880385];
Br J Pharmacol (2005) 146: 744-751 [PMID:16158071]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.