[3H]RS 57639 [Ligand Id: 239] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1908857
  • 5-HT4 receptor in Rat [GtoPdb: 9] [UniProtKB: Q62758]
  • 5-HT4 receptor in Guinea pig [GtoPdb: 9]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT4 receptor in Rat [GtoPdb: 9] [UniProtKB: Q62758]
GtoPdb - - 9.3 pKd - - - Neuropharmacology (1997) 36: 671-9 [PMID:9225293]
5-HT4 receptor in Guinea pig [GtoPdb: 9]
GtoPdb - - 9.7 pKd 0.2 nM Kd Neuropharmacology (1997) 36: 671-9 [PMID:9225293]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]