palmoxiric acid [Ligand Id: 2683] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL12394 (Acide palmoxirique, Acido palmoxirico, MCN-3802, Palmoxiric acid) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| Carnitine palmitoyltransferase 1A in Pig (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2981] [UniProtKB: Q9MYX2] | ||||||||
| ChEMBL | Compound was tested for its inhibitory activity against carnitine palmitoyl transferase-A (CPT-A) | B | 6.05 | pIC50 | 900 | nM | IC50 | J Med Chem (1986) 29: 2184-2190 [PMID:3783579] |
| Carnitine palmitoyltransferase 1A in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3858] [UniProtKB: P32198] | ||||||||
| ChEMBL | Inhibition of carnitine palmitoyl transferase (CPT), assessed with isolated rat liver mitochondria | B | 7.4 | pIC50 | 40 | nM | IC50 | J Med Chem (1987) 30: 1094-1097 [PMID:3585906] |
ChEMBL data shown on this page come from version 34:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
