BAY27-9955 [Ligand Id: 3491] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1933348 (BAY-279955)
  • glucagon receptor/Glucagon receptor in Human [ChEMBL: CHEMBL1985] [GtoPdb: 251] [UniProtKB: P47871]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
glucagon receptor/Glucagon receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1985] [GtoPdb: 251] [UniProtKB: P47871]
ChEMBL Displacement of [125I]Glucagon-Cex from human GCGR B 6.45 pKi 356 nM Ki Bioorg. Med. Chem. Lett. (2012) 22: 415-420 [PMID:22119466]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]