Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
ChEMBL ligand: CHEMBL582985 |
---|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
GPR34 in Human [GtoPdb: 101] [UniProtKB: Q9UPC5] | ||||||||
GtoPdb | - | - | 6.89 | pEC50 | 129 | nM | EC50 |
Biochem Biophys Res Commun (2006) 341: 1078-87 [PMID:16460680]; J Biochem (2012) 151: 511-8 [PMID:22343749] |
GPR34 in Mouse [GtoPdb: 101] [UniProtKB: Q9R1K6] | ||||||||
GtoPdb | - | - | 7.31 | pEC50 | 49 | nM | EC50 | Biochem Biophys Res Commun (2006) 341: 1078-87 [PMID:16460680] |
GPR174 in Human [GtoPdb: 145] [UniProtKB: Q9BXC1] | ||||||||
GtoPdb | - | - | 7.1 | pEC50 | 81 | nM | EC50 | Nat Methods (2012) 9: 1021-9 [PMID:22983457] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]