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ChEMBL ligand: CHEMBL136800 (BDP 12, CX-516, Cx516, BDP-12, CX 516) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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GluA3/GluA4/Glutamate receptor AMPA 3/4 in Rat (target type: PROTEIN COMPLEX) [ChEMBL: CHEMBL3885582] [GtoPdb: 446, 447] [UniProtKB: P19492, P19493] | ||||||||
ChEMBL | Inhibition of GluR3/4 rat in hippocampal neuron | B | 4.02 | pEC50 | 95000 | nM | EC50 | J. Med. Chem. (2010) 53: 7271-7279 [PMID:20839777] |
ChEMBL data shown on this page come from version 27:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]