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ChEMBL ligand: CHEMBL1222250 (Anhydrous dextrose, Anhydrous glucose, Capd, Clintec, Dextro energy, Dextrogel, Dextrose, Dextrose anhydrous, Dextrose, anhydrous, Dextrose solution, Dextrose, unspecified, Dextrose, unspecified form, D-glucose, anhydrous, Gambrosol, Glucose, Glucose-40, Glucose, alpha-d-, Glucose anhydrous, Glucose, anhydrous, Glucose injection, Glucose, liquid, Glucose, unspecified form, Glucosum, anhydrous, Grape sugar, Gsf-syrup, Insta-glucose, Liquid glucose, NSC-406891, Rapilose, Yourgluco) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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Muscle glycogen phosphorylase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3526] [UniProtKB: P11217] | ||||||||
ChEMBL | Inhibitory activity against rabbit muscle glycogen phosphorylase | B | 2.77 | pKi | 2.77 | mM | Log Ki | J Med Chem (1997) 40: 4089-4102 [PMID:9406599] |
ChEMBL data shown on this page come from version 32:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]