α-ketoisocaproate [Ligand Id: 4656] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL445647 (2-Oxoisohexanoate, alpha-Ketoisocaproate, alpha-Oxoisohexanoate)
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Monocarboxylate transporter 2 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2073718] [UniProtKB: Q66HS9]
ChEMBL TP_TRANSPORTER: inhibition of lactate uptake in Xenopus laevis oocytes F 4 pKi 100000 nM Ki Biochem. J. (1999) 341: 529-535 [PMID:10417314]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]