3-hydroxybenzylhydrazine [Ligand Id: 5116] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL352205 (3-Hydrazinomethyl-Phenol) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Gamma-amino-N-butyrate transaminase in Pig (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2266] [UniProtKB: P80147] | ||||||||
| ChEMBL | The Dissociation Constant for Gamma-amino-N-butyrate transaminase | B | 6.34 | pKd | 460 | nM | Kd | J Med Chem (1996) 39: 686-694 [PMID:8576911] |
| ChEMBL | Inhibitory activity against Gamma-amino-N-butyrate transaminase | B | 6.52 | pKi | 300 | nM | Ki | J Med Chem (1996) 39: 686-694 [PMID:8576911] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
