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ChEMBL ligand: CHEMBL574539 (A-804598) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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P2X7/P2X purinoceptor 7 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4805] [GtoPdb: 484] [UniProtKB: Q99572] | ||||||||
ChEMBL | Binding affinity at human P2X7 receptor | B | 8 | pIC50 | 10 | nM | IC50 | Bioorg. Med. Chem. (2009) 17: 4861-4865 [PMID:19540765] |
P2X7/P2X purinoceptor 7 in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5183] [GtoPdb: 484] [UniProtKB: Q9Z1M0] | ||||||||
ChEMBL | Binding affinity at mouse P2X7 receptor | B | 8 | pIC50 | 10 | nM | IC50 | Bioorg. Med. Chem. (2009) 17: 4861-4865 [PMID:19540765] |
P2X7/P2X purinoceptor 7 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2496] [GtoPdb: 484] [UniProtKB: Q64663] | ||||||||
ChEMBL | Binding affinity at rat P2X7 receptor | B | 8 | pIC50 | 10 | nM | IC50 | Bioorg. Med. Chem. (2009) 17: 4861-4865 [PMID:19540765] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]