cilazaprilat [Ligand Id: 6461] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2104578 (Cilazaprilat, Cilazaprilat anhydrous, Cilazapril diacid, RO 31-3113, RO-313113, RO-31-3113)
  • Angiotensin-converting enzyme in Rabbit [GtoPdb: 1613]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Angiotensin-converting enzyme in Rabbit [GtoPdb: 1613]
GtoPdb - - 8.7 pIC50 1.9 nM IC50 Br J Clin Pharmacol (1989) 27 Suppl 2: 139S-150S [PMID:2527528]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]