compound 20 [PMID: 22153340] [Ligand Id: 6568] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1935285
  • MMP12/Matrix metalloproteinase 12 in Human [ChEMBL: CHEMBL4393] [GtoPdb: 1636] [UniProtKB: P39900]
  • This target only has 0 pki data point
  • 0
1 CHEMBL1935285_lig_chart_1 Matrix metalloproteinase 12 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MMP12/Matrix metalloproteinase 12 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4393] [GtoPdb: 1636] [UniProtKB: P39900]
GtoPdb - - 10 pIC50 0.1 nM IC50 Bioorg Med Chem Lett (2012) 22: 138-43 [PMID:22153340]
ChEMBL Inhibition of human MMP-12 B 10 pIC50 0.1 nM IC50 Bioorg. Med. Chem. Lett. (2012) 22: 138-143 [PMID:22153340]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]