pemirolast [Ligand Id: 7329] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1201198 (Pemirolast)
  • GPR35/G protein-coupled receptor GPR35 in Rat [ChEMBL: CHEMBL2390812] [GtoPdb: 102] [UniProtKB: Q33BM1]
  • This target only has 0 pki data point
  • 0
1 CHEMBL1201198_lig_chart_1 G protein-coupled receptor GPR35 Rat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GPR35/G protein-coupled receptor GPR35 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2390812] [GtoPdb: 102] [UniProtKB: Q33BM1]
ChEMBL Agonist activity at recombinant rat N-terminal FLAG/eYFP-fused GPR35 expressed in HEK293 cells assessed as induction of beta-arrestin recruitment by BRET assay F 7.02 pEC50 95 nM EC50 ACS Med Chem Lett (2018) 9: 422-427 [PMID:29795753]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]