etazolate [Ligand Id: 7336] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL356388 (EHT-0202, Etazolate, SQ-20009)
  • GABAA receptor β3 subunit in Human [GtoPdb: 412] [UniProtKB: P28472]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GABAA receptor β3 subunit in Human [GtoPdb: 412] [UniProtKB: P28472]
GtoPdb inhibition of [35S]TBPS binding - 5.46 pIC50 3500 nM IC50 Eur J Pharmacol (1996) 301: 207-14 [PMID:8773466]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]