compound 1 [PMID: 15724976] [Ligand Id: 7507] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL3220205
  • lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
GtoPdb ELISA assay measuring binding to the KAT2B (PCAF) bromodomain (GST-tagged protein containing amino acid residues 719-832) . - 8.29 pIC50 5.1 nM IC50 J Am Chem Soc (2005) 127: 2376-7 [PMID:15724976]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]