compound 1 [PMID: 15724976] [Ligand Id: 7507] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL3220205 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831] | ||||||||
| GtoPdb | ELISA assay measuring binding to the KAT2B (PCAF) bromodomain (GST-tagged protein containing amino acid residues 719-832) . | - | 8.29 | pIC50 | 5.1 | nM | IC50 | J Am Chem Soc (2005) 127: 2376-7 [PMID:15724976] |
ChEMBL data shown on this page come from version 28:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]
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