ChEMBL ligand: CHEMBL1236441
CREB binding protein/CREB-binding protein in Human [ChEMBL: CHEMBL5747] [GtoPdb: 2734] [UniProtKB: Q92793] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
CREB binding protein/CREB-binding protein in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5747] [GtoPdb: 2734] [UniProtKB: Q92793]
ChEMBL	Displacement of biotinylated p53-AcK382 from GST-tagged CREBBP (1082 to 1197 amino acid residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells by tryptophan fluorescence assay	B	4.7	pKd	20000	nM	Kd	Medchemcomm (2015) 6: 1587-1604
ChEMBL	Binding affinity to CBP bromodomain (unknown origin) by fluorescence spectroscopic analysis	B	4.71	pKd	19600	nM	Kd	J Med Chem (2016) 59: 1271-1298 [PMID:26572217]
ChEMBL	Inhibition of N-terminally biotinylated p53 AcK382 peptide binding to GST-fused CBP bromodomain (1082 to 1197) (unknown origin) expressed in Escherichia coli by Western blot analysis	B	4.71	pKd	19600	nM	Kd	Medchemcomm (2016) 7: 2246-2264 [PMID:29170712]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]